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16 p, 3.1 MB Neuroprotective effects of the multitarget agent AVCRI104P3 in brain of middle-aged mice / Relat Pardo, Júlia (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ; Come, Julio (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ; Pérez, Belén (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ; Camps-Renom, Pol (Universitat de Barcelona. Institut de Biomedicina) ; Muñoz-Torrero López-Ibarra, Diego (Universitat de Barcelona. Institut de Biomedicina) ; Badía, A. (Albert) (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ; Gimenez-Llort, Lydia (Universitat Autònoma de Barcelona. Departament de Psiquiatria i de Medicina Legal) ; Clos, M. Victoria (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia)
Molecular factors involved in neuroprotection are key in the design of novel multitarget drugs in aging and neurodegeneration. AVCRI104P3 is a huprine derivative that exhibits potent inhibitory effects on human AChE, BuChE, and BACE-1 activities, as well as on AChE-induced and self-induced Aβ aggregation. [...]
2018 - 10.3390/ijms19092615
International journal of molecular sciences, Vol. 19 Núm. 9 (april 2018) , p. 2615  

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1 Come, Julio
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