1.
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19 p, 765.0 KB |
Abuse Potential of Cathinones in Humans : a Systematic Review
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Poyatos, Lourdes (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Torres, Adrian (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Papaseit, Esther (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Pérez-Mañá, Clara (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Hladun, Olga (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Núñez-Montero, Melani (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
de la Rosa, Georgina (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Torrens, Marta (Universitat Autònoma de Barcelona. Departament de Psiquiatria i de Medicina Legal) ;
Fuster, Daniel (Universitat Autònoma de Barcelona. Departament de Medicina) ;
Muga, Roberto (Universitat Autònoma de Barcelona. Departament de Medicina) ;
Farre, Magi (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia)
Introduction and objective: Assessing the abuse potential of new substances with central nervous system activity is essential for preventing possible risks of misuse and addiction. The same methodology is recommended for the evaluation of the abuse potential of recreational drugs. [...]
2022 - 10.3390/jcm11041004
Journal of clinical medicine, Vol. 11 Núm. 4 (february 2022) , p. 1004
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2.
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14 p, 1.2 MB |
Daidzein modulates cocaine-reinforcing effects and cue-induced cocaine reinstatement in CD-1 male mice
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Martin, Miquel (Universitat Pompeu Fabra. Parc de Recerca Biomèdica de Barcelona) ;
Gutiérrez-Martos, Miriam (Universitat Pompeu Fabra.Parc de Recerca Biomèdica de Barcelona) ;
Cabrera, Roberto (Universitat Pompeu Fabra. Parc de Recerca Biomèdica de Barcelona) ;
Langohr, Klaus (Universitat Politècnica de Catalunya. Departament d'Estadística i Investigació Operativa) ;
Maldonado, Rafael (Universitat Pompeu Fabra) ;
Farre, Magi (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
de la Torre, Rafael (Universitat Pompeu Fabra) ;
Universitat Autònoma de Barcelona
Cocaine addiction is a chronic relapsing disorder that lacks of an effective treatment. Isoflavones are a family of compounds present in different plants and vegetables like soybeans that share a common chemical structure. [...]
2021 - 10.1007/s00213-021-05820-z
Psychopharmacology, Vol. 238 (april 2021) , p. 1923-1936
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3.
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14 p, 991.2 KB |
Acute Pharmacological Effects and Oral Fluid Biomarkers of the Synthetic Cannabinoid UR-144 and THC in Recreational Users
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Maida, Nunzia La (Università Politecnica delle Marche (Ancona, Itàlia). Department of Excellence of Biomedical Science and Public Health) ;
Papaseit, Esther (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Martínez, Lucia (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Pérez-Mañá, Clara (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Poyatos, Lourdes (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Pellegrini, Manuela (Istituto Superiore di Sanità (Roma, Itàlia). National Centre on Addiction and Doping) ;
Pichini, Simona (Istituto Superiore di Sanità (Roma, Itàlia). National Centre on Addiction and Doping) ;
Pacifici, Roberta (Istituto Superiore di Sanità (Roma, Itàlia). National Centre on Addiction and Doping) ;
Ventura, Mireia (Associació Benestar i Desenvolupament (Barcelona)) ;
Galindo, Liliana (Associació Benestar i Desenvolupament (Barcelona)) ;
Busardò, Francesco Paolo (Università Politecnica delle Marche (Ancona, Itàlia). Department of Excellence of Biomedical Science and Public Health) ;
Farre, Magi (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia)
UR-144 is a synthetic cannabinoid found in herbal incenses for recreational use as a substitute of cannabis. It is a cannabinoid receptor agonist with effects on the central nervous system similar to those of THC. [...]
2021 - 10.3390/biology10040257
Biology, Vol. 10 Núm. 4 (march 2021)
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4.
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9 p, 999.0 KB |
Long-Term Outcomes of Patients With Cocaine Use Disorder : A 18-years Addiction Cohort Study
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Sanvisens, Arantza (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Hernandez-Rubio, Anna (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Zuluaga Cruz, Andrea Paola (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Fuster, Daniel (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Papaseit, Esther (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Galan, Sara (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Farre, Magi (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Muga, Roberto (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Universitat Autònoma de Barcelona
Objective: Cocaine Use Disorder (CUD) has been associated with multiple complications and premature death. The purpose of the present study was to analyze the relationship between baseline medical comorbidity and long-term medical outcomes (i. [...]
2021 - 10.3389/fphar.2021.625610
Frontiers in Pharmacology, Vol. 12 (february 2021)
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5.
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13 p, 1013.2 KB |
Acute Pharmacological Effects of Oral and Intranasal Mephedrone : an observational study in humans
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Papaseit, Esther (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Olesti, Eulàlia (Universitat Pompeu Fabra. Grup de Recerca en Farmacologia i Neurociències) ;
Pérez-Mañá, Clara (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Torrens, Marta (Universitat Autònoma de Barcelona. Departament de Psiquiatria i de Medicina Legal) ;
Fonseca, Francina (Universitat Autònoma de Barcelona. Departament de Psiquiatria i de Medicina Legal) ;
Grifell, Marc (Universitat Autònoma de Barcelona. Departament de Psiquiatria i de Medicina Legal) ;
Ventura, Mireia (Associació Benestar i Desenvolupament) ;
de la Torre, Rafael (Institut Hospital del Mar d'Investigacions Mèdiques) ;
Farre, Magi (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia)
Mephedrone (4-methylmethcathinone) is a synthetic cathinone with psychostimulant properties which remains one of the most popular new psychoactive substances (NPS). It is frequently used orally and/or intranasally. [...]
2021 - 10.3390/ph14020100
Pharmaceuticals, Vol. 14 Núm. 2 (2021) , p. 100
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14 p, 1.5 MB |
Disposition of Phytocannabinoids, Their Acidic Precursors and Their Metabolites in Biological Matrices of Healthy Individuals Treated with Vaporized Medical Cannabis
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Busardò, Francesco Paolo (Department of Excellence-Biomedical Sciences and Public Health, Università Politecnica delle Marche, 60121 Ancona, Italy) ;
Pérez-Acevedo, Ana Pilar (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Pacifici, Roberta (National Centre on Addiction and Doping, Istituto Superiore di Sanità, 00161 Rome, Italy) ;
Mannocchi, Giulio (School of Law, University of Camerino, 62032 Camerino, Italy) ;
Gottardi, Massimo (Comedical S.Rl, 38123 Trento, Italy) ;
Papaseit, Esther (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Pérez-Mañá, Clara (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Martin, Soraya (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Poyatos, Lourdes (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Pichini, Simona (National Centre on Addiction and Doping, Istituto Superiore di Sanità, 00161 Rome, Italy) ;
Farre, Magi (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia)
Inhalation by vaporization is a useful application mode for medical cannabis. In this study, we present the disposition of Δ9-tetrahydrocannabinol (THC), cannabidiol (CBD), their acidic precursors, and their metabolites in serum, oral fluid, and urine together with the acute pharmacological effects in 14 healthy individuals treated with vaporized medical cannabis. [...]
2021 - 10.3390/ph14010059
Pharmaceuticals, Vol. 14 (january 2021)
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7.
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21 p, 893.8 KB |
Oral Administration of Cannabis and Δ-9-tetrahydrocannabinol (THC) Preparations : A Systematic Review
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Poyatos, Lourdes (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Pérez-Acevedo, Ana Pilar (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Papaseit, Esther (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Pérez Mañá, Clara (Institut Germans Trias i Pujol) ;
Martin, Soraya (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Hladun, Olga (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Siles, Adrià (Institut Germans Trias i Pujol) ;
Torrens, Marta (Universitat Autònoma de Barcelona. Departament de Psiquiatria i de Medicina Legal) ;
Busardo, Francesco Paolo (Università Politecnica delle Marche, Ancona) ;
Farre, Magi (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol)
Background and objective : Changes in cannabis legalization regimes in several countries have influenced the diversification of cannabis use. There is an ever-increasing number of cannabis forms available, which are gaining popularity for both recreational and therapeutic use. [...]
2020 - 10.3390/medicina56060309
Medicina, Vol. 56 (june 2020)
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10 p, 328.8 KB |
Cannabinoids : from pot to lab
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Papaseit, Esther (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Pérez-Mañá, Clara (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Pérez-Acevedo, Ana Pilar (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Hladun, Olga (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Torres-Moreno, M. Carmen (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Muga, Roberto (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Torrens, Marta (Universitat Autònoma de Barcelona. Departament de Psiquiatria i de Medicina Legal) ;
Farre, Magi (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia)
Cannabis is becoming increasingly present in our society. In recent years, the line between the natural (cannabis) and the synthetic (synthetic cannabinoids), the recreational (cannabis) and the medical (pharmaceutical cannabinoids and medical cannabis) has been crossed. [...]
2018 - 10.7150/ijms.27087
International Journal of Medical Sciences, Vol. 15 (august 2018) , p. 1286-1295
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13 p, 839.9 KB |
Acute Effects of 2C-E in Humans : An Observational Study
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Papaseit, Esther (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Olesti, Eulàlia (Universitat Pompeu Fabra. Departament de Ciències Experimentals i de la Salut) ;
Pérez-Mañá, Clara (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia) ;
Torrens, Marta (Drug Addiction Program, Institut de Neuropsiquiatria i Adiccions (INAD)) ;
Grifell, Marc (Energy Control, Associació Benestar i Desenvolupament) ;
Ventura, Mireia (Energy Control, Associació Benestar i Desenvolupament) ;
Pozo, Oscar J. (Institut Hospital del Mar d'Investigacions Mèdiques) ;
de Sousa Fernandes Perna, Elizabeth B. (Maastricht University. Department of Neuropsychology and Psychopharmacology) ;
Ramaekers, Johannes G. (Maastricht University. Department of Neuropsychology and Psychopharmacology) ;
de la Torre, Rafael (Universitat Pompeu Fabra. Departament de Ciències Experimentals i de la Salut) ;
Farre, Magi (Universitat Autònoma de Barcelona. Departament de Farmacologia, de Terapèutica i de Toxicologia)
2,5-Dimethoxy-4-ethylphenethylamine (2C-E) is psychedelic phenylethylamine, with a chemical structure similar to mescaline, used as new psychoactive substance (NPS). It inhibits norepinephrine and serotonin uptake and, more relevant, acts as a partial agonist of the serotonin 2A (5-HT), 2B (5-HT), and (5-HT) receptors. [...]
2020 - 10.3389/fphar.2020.00233
Frontiers in Pharmacology, Vol. 11 (march 2020)
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10.
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9 p, 287.3 KB |
Psychopathological symptoms associated with synthetic cannabinoid use : a comparison with natural cannabis
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Mensen, Vincent T. (Department of Drug Monitoring, Utrecht, The Netherlands) ;
Vreeker, Annabel (University of Utrecht. University Medical Center Utrecht, Department of Psychiatry) ;
Nordgren, Johan (Malmö University. Department of Social Work) ;
Atkinson, Amanda (Liverpool John Moores University. Public Health Institute) ;
de la Torre, Rafael (Institut Hospital del Mar d'Investigacions Mèdiques) ;
Farre, Magi (Institut Germans Trias i Pujol. Hospital Universitari Germans Trias i Pujol) ;
Ramaekers, Johannes G. (Maastricht University. Department of Neuropsychology and Psychopharmacology, Faculty of Psychology and Neuroscience) ;
Brunt, Tibor M. (Radboud University. Department of Developmental Psychopathology) ;
Universitat Autònoma de Barcelona
Synthetic cannabinoids (SCs) are a class of new psychoactive substances that have been rapidly evolving around the world throughout recent years. Many different synthetic cannabinoid analogues are on the consumer market and sold under misleading names, like "spice" or "incense. [...]
2019 - 10.1007/s00213-019-05238-8
Psychopharmacology, Vol. 236 (april 2019) , p. 2677-2685
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