Dipòsit Digital de Documents de la UAB 2 registres trobats  La cerca s'ha fet en 0.00 segons. 
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11 p, 1.8 MB A Complementary Scale of Biased Agonism for Agonists with Differing Maximal Responses / Burgueño, Javier (Department of Pharmacology, Drug Discovery & Preclinical Development, ESTEVE) ; Pujol Argemí, Marta (Department of Pharmacology, Drug Discovery & Preclinical Development, ESTEVE) ; Monroy, Xavier (Department of Pharmacology, Drug Discovery & Preclinical Development, ESTEVE) ; Roche, David (Universitat Internacional de Catalunya. Facultat de Ciències Econòmiques i Socials) ; Varela, Maria Jose (Universidade de Santiago de Compostela) ; Merlos, Manuel (Department of Pharmacology, Drug Discovery & Preclinical Development, ESTEVE) ; Giraldo, Jesús (Universitat Autònoma de Barcelona. Institut de Neurociències) ; Universitat Autònoma de Barcelona. Departament de Pediatria, Obstetrícia i Ginecologia i de Medicina Preventiva i Salut Pública
Compelling data in the literature from the recent years leave no doubt about the pluridimensional nature of G protein-coupled receptor function and the fact that some ligands can couple with different efficacies to the multiple pathways that a receptor can signal through, a phenomenon most commonly known as functional selectivity or biased agonism. [...]
2017 - 10.1038/s41598-017-15258-z
Scientific reports, Vol. 7 (november 2017)  
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17 p, 2.9 MB Analysis of Human Dopamine D Receptor Quaternary Structure / Marsango, Sara (University of Glasgow) ; Caltabiano, Gianluigi 1978- (Universitat Autònoma de Barcelona. Laboratori de Medicina Computacional) ; Pou, Chantevy (University of Glasgow) ; Varela Liste, María José (University of Glasgow) ; Milligan, Graeme (University of Glasgow)
Background: The dopamine D receptor can form dimers/oligomers, but the molecular basis for this is poorly defined. Results: Molecular modeling, mutagenesis, and analysis of inactive state receptor crystal structures allowed assessment of models of receptor organization. [...]
2015 - 10.1074/jbc.M114.630681
Journal of biological chemistry, Vol. 290 (april 2015) , p. 15146-15162  

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