Resultats globals: 2 registres trobats en 0.02 segons.
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18 p, 1.7 MB Essential Control of the Function of the Striatopallidal Neuron by Pre-coupled Complexes of Adenosine A-Dopamine D Receptor Heterotetramers and Adenylyl Cyclase / Ferré, Sergi (National Institutes of Health, Baltimore, United States) ; Bonaventura, Jordi (National Institutes of Health, Baltimore, United States) ; Zhu, Wendy (Circuit Therapeutics, Menlo Park, United States) ; Hatcher-Solis, Candice (National Institutes of Health, Baltimore, United States) ; Taura, Jaume (Universitat de Barcelona. Institut de Neurociències) ; Quiroz, César (National Institutes of Health, Baltimore, United States) ; Cai, Ning-Sheng (National Institutes of Health, Baltimore, United States) ; Moreno, Estefanía (Universitat de Barcelona. Departament de Bioquímica i Biomedicina Molecular) ; Casadó-Anguera, Verònica (Universitat de Barcelona. Departament de Bioquímica i Biomedicina Molecular) ; Kravitz, Alexxai V. (National Institutes of Health, Bethesda, United States) ; Thompson, Kimberly R. (Circuit Therapeutics, Inc., Menlo Park, United States) ; Tomasi, Dardo G. (National Institutes of Health, Rockville, United States) ; Navarro Brugal, Gemma (Universitat de Barcelona. Departament de Bioquímica i Fisiologia) ; Cordomí Montoya, Arnau (Universitat Autònoma de Barcelona. Laboratori de Medicina Computacional) ; Pardo Carrasco, Leonardo (Universitat Autònoma de Barcelona. Laboratori de Medicina Computacional) ; Lluís, Carme (Universitat de Barcelona. Departament de Bioquímica i Biomedicina Molecular) ; Dessauer, Carmen W. (University of Texas Health Science Center at Houston, United States) ; Volkow, Nora D. (National Institutes of Health, Rockville, United States) ; Casadó, Vicent (Universitat de Barcelona. Departament de Bioquímica i Biomedicina Molecular) ; Ciruela, Francisco (Universitat de Barcelona. Institut de Neurociències) ; Logothetis, Diomedes E. (Northeastern University, Boston, United States) ; Zwilling, Daniel (Circuit Therapeutics, Inc, Menlo Park, United States)
The central adenosine system and adenosine receptors play a fundamental role in the modulation of dopaminergic neurotransmission. This is mostly achieved by the strategic co-localization of different adenosine and dopamine receptor subtypes in the two populations of striatal efferent neurons, striatonigral and striatopallidal, that give rise to the direct and indirect striatal efferent pathways, respectively. [...]
2018 - 10.3389/fphar.2018.00243
Frontiers in Pharmacology, Vol. 9 (april 2018)  

Documents de recerca 1 registres trobats  
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21 p, 2.0 MB Unique pharmacodynamic properties and low abuse liability of the μ-opioid receptor ligand (S)-methadone / Michaelides, Michael (NIH) ; Levinstein, Marjorie (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; De Oliveira, Paulo (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; Casajuana-Martin, Nil (Universitat Autònoma de Barcelona) ; Quiroz, Cesar (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; Budinich, Reece (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; Rais, Rana (Johns Hopkins School of Medicine) ; Rea, William (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; Ventriglia, Emilya (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; Llopart, Natàlia (Universitat de Barcelona) ; Casadó-Anguera, Verònica (Universitat de Barcelona) ; Moreno, Estefanía (University of Barcelona. Department of Biochemistry and Molecular Biomedicine) ; Walther, Donna (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; Glatfelter, Grant (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; Weinshenker, David ; Zarate, Carlos (NIMH) ; Casadó, Vicent (Universitat de Barcelona) ; Baumann, Michael (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica)) ; Pardo Carrasco, Leonardo (Universitat Autònoma de Barcelona) ; Ferré, Sergi (National Institute on Drug Abuse (Baltimore, Estats Units d'Amèrica))
(R,S)-methadone ((R,S)-MTD) is a racemic μ-opioid receptor (MOR) agonist comprised of (R)-MTD and (S)-MTD enantiomers used for the treatment of opioid use disorder (OUD) and pain. (R)-MTD is used as an OUD treatment, has high MOR potency, and is believed to mediate (R,S)-MTD's therapeutic efficacy. [...]
2023 - 10.21203/rs.3.rs-2644719/v1  

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2 Quiroz, César
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