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14 p, 14.9 MB Repurposing Itraconazole and Hydroxychloroquine to Target Lysosomal Homeostasis in Epithelial Ovarian Cancer / Marastoni, Stefano (University Health Network (Canadà)) ; Madariaga, Ainhoa (Universitat Autònoma de Barcelona) ; Pesic, Aleksandra (University Health Network (Canada)) ; Nair, Sree Narayanan (University Health Network (Canada)) ; Li, Zhu Juan (University Health Network (Canada)) ; Shalev, Zvi (University Health Network (Canada)) ; Ketela, Troy (University Health Network (Canada)) ; Colombo, Ilaria (University Health Network (Canada)) ; Mandilaras, Victoria (University Health Network (Canada)) ; Cabanero, Michael (University Health Network (Canada)) ; Bruce, Jeff P. (University Health Network (Canada)) ; Li, Xuan (University Health Network (Canada)) ; Garg, Swati (University Health Network (Canada)) ; Wang, Lisa (University Health Network (Canada)) ; Chen, Eric X. (University Health Network (Canada)) ; Gill, Sarbjot (University Health Network (Canada)) ; Dhani, Neesha C. (University Health Network (Canada)) ; Zhang, Wenjiang (University Health Network (Canada)) ; Pintilie, Melania (University Health Network (Canada)) ; Bowering, Valerie (University Health Network (Canada)) ; Koritzinsky, Marianne (University Health Network (Canada)) ; Rottapel, Robert (University Health Network (Canada)) ; Wouters, Bradly G. (Department of Radiation Oncology, University of Toronto) ; Oza, Amit M. (University Health Network (Canada)) ; Joshua, Anthony M. (Garvan Institute of Medical Research (Austràlia)) ; Lheureux, Stephanie (Princess Margaret Cancer Centre)
The combination of the antifungal drug itraconazole with antimalarial drug hydroxychloroquine leads to a cytotoxic lysosomal dysfunction, supporting the rational for further research on lysosomal targeting in ovarian cancer.
2022 - 10.1158/2767-9764.CRC-22-0037
Cancer Research Communications, Vol. 2 (may 2022) , p. 293-306  

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