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6 p, 2.3 MB Bioconjugated technetium carbonyls by transmetalation reaction with zinc derivatives / Borràs, Jordi (Universitat Autònoma de Barcelona. Departament de Química) ; Lecina Vicente, Joan (Universitat Autònoma de Barcelona. Departament de Química) ; Foster, Julie (Queen Mary University of London. John Vane Science Centre) ; Kashani, Roxana (Queen Mary University of London. John Vane Science Centre) ; Melendez-Alafort, L. (Istituto Oncologico Veneto IRCCS) ; Sosabowski, Jane (Queen Mary University of London. John Vane Science Centre) ; Suades Ortuño, Joan (Universitat Autònoma de Barcelona. Departament de Química)
The transmetalation reaction between zinc dithiocarbamates functionalized with organic groups and the cation fac-[Tc(HO)(CO)] has been studied as a new strategy to bind biomolecules to this radionuclide for preparing radiopharmaceuticals with high molar activity. [...]
2021 - 10.1016/j.bmcl.2021.127840
Bioorganic and Medicinal Chemistry Letters, Vol. 37 (April 2021) , art. 127840  

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