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17 p, 4.4 MB Perspective on the structural basis for human aldo-keto reductase 1b10 inhibition / Ruiz, Francesc Xavier (Rutgers University. Department of Chemistry and Chemical Biology) ; Parés i Casasampera, Xavier (Universitat Autònoma de Barcelona. Departament de Bioquímica i de Biologia Molecular) ; Farrés, Jaume (Universitat Autònoma de Barcelona. Departament de Bioquímica i de Biologia Molecular)
Human aldo-keto reductase 1B10 (AKR1B10) is overexpressed in many cancer types and is involved in chemoresistance. This makes AKR1B10 to be an interesting drug target and thus many enzyme inhibitors have been investigated. [...]
2021 - 10.3390/metabo11120865
Metabolites, Vol. 11, Issue 12 (December 2021) , art. 865  

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